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Amino Tadalafil poda mugadziri CAS Nha.: 385769-84-6 98% kuchena min.zvekuwedzera zvinhu

Tsanangudzo Pfupi

Amino Tadalafil isanganiswa yakafanana neTadalafil, ine mamwe emapoka anoshanda muchimiro chayo achitsiviwa nemapoka emamino.


Product Detail

Product Tags

Product Parameters

Product name

Amino Tadalafil

Rimwe zita

(6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[ 3,4-b]indole-1,4-dione;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A -Hexahydropyrazino[1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dione;(6R,12aR)-2-Amino-6-(benzo[d][1,3] ]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R ,12aR) -2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3] ,4-b]indole-1,4(6H,7H)-dione

CAS Nha.

385769-84-6

Molecular formula

C21H18N4O4

Molecular uremu

390.39

Kuchena

98.0%

Chitarisiko

Hupfu hwakachena kusvika kuchena

Application

Dietary Supplement Raw Material

Product sumo

Amino Tadalafil isanganiswa yakafanana neTadalafil, ine mamwe emapoka anoshanda muchimiro chayo achitsiviwa nemapoka emamino.Iyo PDE5 inhibitor uye ine pharmacological mhedzisiro yakafanana neTadalafil.Inonyanya kushandiswa pakurapa kwemurume erectile dysfunction (ED).Kuenzaniswa neTadalafil, Amino Tadalafil ine chiyero chinononoka chemetabolism mumuviri, uye nekudaro inogona kuva nemhedzisiro inogara kwenguva refu.

Feature

(1) High selectivity: Amino Tadalafil ine high selectivity ye PDE5, ine hukama hwepamusoro hwePDE5 kupfuura dzimwe PDE subtypes.Izvi zvinoreva kuti Amino Tadalafil inogona kunyatsovhara basa rePDE5 enzyme, kukurudzira kuyerera kweropa munhengo dzekubereka dzechirume uye nekuvandudza zviratidzo zve erectile dysfunction (ED).

(2) Inogara kwenguva refu: Amino Tadalafil ine inononoka metabolism rate mumuviri, iyo inobvumira kuti ibudise yakawedzera kwenguva yakareba pharmacological effect, inogara kusvika kumaawa 36.Izvi zvinoita kuti Amino Tadalafil ave akareba-anoita ED kurapwa mushonga, izvo zvisingadi kutorwa kazhinji.

(3) Zvishoma zvinokonzerwa nemigumisiro: Amino Tadalafil ine zvishoma zvinokonzerwa neTadalafil, zvakadai semusoro, uye kusagadzikana kwepamuviri.Nekuda kwekusarudzwa kwayo kwepamusoro, Amino Tadalafil inogona kunyatso dzivirira kusangana nemamwe maPDE subtypes, kuderedza chiitiko chemhedzisiro.

(4) Wide application tarisiro: Pamusoro pekurapa ED, Amino Tadalafil inogona zvakare kushandiswa kurapa zvimwe zvirwere senge pulmonary arterial hypertension.Izvi zvinoita kuti Amino Tadalafil ave netarisiro yakakura yekushandisa mune ramangwana.

Applications

Amino Tadalafil musanganiswa wakagadzirwa mumakore achangopfuura, ane chimiro chakafanana neTadalafil, asi mamwe mapoka muchimiro chayo anotsiviwa nemapoka emamino.Parizvino, Amino Tadalafil haisati yatenderwa kuti ishandiswe pakurapa, saka kushanda kwayo mundima yekurapa ishoma.Nekudaro, zvimwe zvidzidzo zvakaratidza kuti komboni iyi ine mukana mukuru wekushandisa.

Amino Tadalafil ndeye PDE5 inhibitor, iyo ine yakafanana pharmacological effect seTadalafil.Inogona kuvandudza zviratidzo zve erectile dysfunction (ED) nekusimudzira kuyerera kweropa munhengo dzechirume dzekubereka nekuvhara basa rePDE5 enzyme.Kuenzaniswa neTadalafil, Amino Tadalafil ine inononoka metabolism rate mumuviri, iyo inogona kuva nemhedzisiro inogara.Izvi zvinoita kuti Amino Tadalafil ave nekugona kukuru mukurapa kweED.

Pamusoro pezvo, Amino Tadalafil inogona zvakare kushandiswa kurapa zvimwe zvirwere, senge pulmonary arterial hypertension.Zvimwe zvidzidzo zvakaratidza kuti PDE5 inhibitors inogona kuderedza mitsipa yeropa, nekudaro inovandudza zviratidzo zvevarwere vane pulmonary arterial hypertension.Nekuti Amino Tadalafil ine yakafanana pharmacological mhedzisiro seTadalafil, inogona zvakare kushandiswa kurapa pulmonary arterial hypertension.

Pakazere, Amino Tadalafil ine mukana mukuru wekushandisa, asi mimwe miedzo yekiriniki inodiwa kuti uone kuchengetedzeka kwayo uye kushanda kwayo.Kana iyi miedzo ikaunza mhedzisiro yakanaka, Amino Tadalafil inogona kuve mushonga mutsva wekurapa ED uye pulmonary arterial hypertension, ichipa mamwe marapirwo emakiriniki vanachiremba nevarwere.


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