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Coluracetam poda mugadziri CAS Nha.: 135463-81-9 99% kuchena min.zvekuwedzera zvinhu

Tsanangudzo Pfupi

Coluracetam inhengo yemhuri ye racetam ye nootropic compounds uye inonziwo MKC-231.Yakagadzirwa neKobe Pharmaceutical Company muJapan nechinangwa chekurapa AD nekushaya njere.


Product Detail

Product Tags

Product Parameters

Product name

Coluracetam

Rimwe zita

MKC-231;

2-oxo-N-(5,6,7,8-tetrahydro-2,3-dimethyl-furo[2,3-b]quinolin-4-yl) -1-pyrrolidineacetamide

CAS Nha.

135463-81-9

Molecular formula

C19H23N3O3

Molecular uremu

341.4

Kuchena

99.0%

Chitarisiko

Upfu chena

Application

Dietary Supplement Raw Material

Product sumo

Coluracetam inhengo yemhuri ye racetam ye nootropic compounds uye inonziwo MKC-231.Yakagadzirwa neKobe Pharmaceutical Company muJapan nechinangwa chekurapa AD nekushaya njere.

Iyo chaiyo nzira yekuita kweColuracetam haina kunyatsonzwisiswa, asi inotendwa kuti inonyanya kushanda nekugadzirisa cholinergic system.Inofungidzirwa kuwedzera mazinga eacetylcholine, inokosha neurotransmitter muuropi iyo yakanyatsobatanidzwa nekudzidza nekuyeuka mabasa.Coluracetam inogona kuita izvi nekuwedzera nhamba uye basa recholine uptake transporters, zvichiita kuti kuwedzerwa kusunungurwa kweacetylcholine uye kuwedzerwa kwechiratidzo chekufambisa pakati peeuroni.

Kunyange zvazvo tsvakurudzo yeColuracetam ichiri shoma, kumwe kuedza kwepakutanga uye zvidzidzo zvemhuka zvakaratidza zvinogona kuitika neuroprotective uye cognitive-enhancing effects.Zvimwe zvidzidzo zvakawana kuti Coluracetam ine imwe gadziriso mukukanganisika kwendangariro mumhando dzeAD.

Maererano nekutsvakurudza kwekliniki, zvidzidzo zveColuracetam zvakanyanyotarisa pakuedza kwemhuka uye miedzo yepakutanga yevanhu.Kutsvakurudza kwakawanda uye humbowo hunodiwa kuti uone kuchengetedzeka kwayo uye kushanda kwayo muvanhu.Parizvino, Coluracetam haina kubvumirwa kushandiswa kwekliniki, asi inoshandiswa zvakanyanya sekuwedzera kwenootropic yekuvandudza ruzivo mune dzimwe nyika.

Nezve kuchengeteka, pane zvishoma zvinyorwa zvekutsvakurudza zvinowanikwa pamigumisiro yemigumisiro uye njodzi dzenguva refu dzeColuracetam.Kubva pane ruzivo rwezvino, Coluracetam inowanzoonekwa seyakachengeteka, asi ichiri kukurudzirwa kutaurirana nenyanzvi yezvehutano, kunyanya kana iwe uine chero mamiriro ehutano kana uri kutora mimwe mishonga, usati waishandisa.

Muchidimbu, Coluracetam inhengo ye nootropic iyo iri kuongororwa nokuda kwekugona kwayo mukurapa AD uye kukanganisa kwekuziva.Nepo kumwe kutsvagurudza kwekutanga kunoratidza kuwedzeredzwa kwekuziva uye neuroprotective mhedzisiro, zvimwe zvidzidzo zvinodikanwa kumisikidza kushanda kwayo kwechokwadi uye kuchengetedzeka.

Feature

(1) Kuchena Kwakakwirira: Coluracetam inogadzirirwa kushandiswa kwepamusoro uye maitiro ekugadzira, kuve nechokwadi chepamusoro chekuchena.Uku kuchena kwepamusoro kunobatsira kuvandudza bioavailability uye kunoderedza kuitika kweakaipa maitiro.

(2) Kuchengetedza: Coluracetam inonzi yakachengeteka kuti ishandiswe nevanhu.Zvidzidzo zvakakura zvakaratidza kuderera kwayo muchetura uye kushoma mhedzisiro mukati meiyo yakakurudzirwa dosi renji.

(3) Kugadzikana: Kugadzirira kweColuracetam kunoratidza kugadzikana kwakanakisisa, kuchengetedza basa ravo uye kubudirira pasi pemamiriro akasiyana-siyana ezvakatipoteredza nekuchengetedza.Uku kugadzikana kunovimbisa kuenderana uye kwakavimbika kuita nekufamba kwenguva.

(4) Rapid Absorption: Coluracetam inotorwa nyore nyore nemuviri wemunhu.Pakunwa, inokurumidza kupinda muropa kuburikidza nemukati wemukati uye inonyatsogovera kune zvakasiyana-siyana uye nhengo, zvichiita kuti iite zvaanoda.

(5) Cognitive Enhancement: Coluracetam inozivikanwa nokuda kwekukwanisa kwayo kuwedzera basa rekuziva, kusanganisira kuvandudzwa kwekuyeuka, kukwanisa kudzidza, uye kutarisa.Inowanzotsvakwa nevanhu vari kutsvaga kukwenenzvera kuita kwavo pfungwa.

(6) Neuroprotective Effects: Tsvagiridzo inoratidza kuti Coluracetam inogona kuve neuroprotective zvimiro, izvo zvinogona kubatsira kuchengetedza kubva kune zera-ane hukama kuderera kwekuziva uye kutsigira hutano hwehuropi hwese.

(7) Inogona Kurapa Kushungurudzika Kwepfungwa: Coluracetam inoratidza chivimbiso sechingangove chekurapa sarudzo yekusagadzikana kwepfungwa, senge Alzheimer's disease uye mamwe neurodegenerative mamiriro.Zvisinei, kumwe kutsvakurudza kunodiwa kuti unzwisise zvizere kushanda kwayo mukurapa aya chaiwo mamiriro.

Applications

Coluracetam parizvino iri kushandiswa mumhando dzakasiyana siyana uye inoratidza tarisiro inovimbisa yeramangwana.Inonyanya kushandiswa seyekuwedzera yekuziva yekuwedzera, inotsvakwa nevanhu vanotarisa kuvandudza ndangariro, kutarisa, uye kugona kudzidza.Iko kugona kwekomboni kugadzirisa iyo cholinergic system inotendwa kuti inobatsira kune yayo yekuziva-inosimudzira mhedzisiro.

Pamusoro pemashandisirwo ayo azvino, Coluracetam yakaratidza kugona mukurapa neurodegenerative kusagadzikana senge Alzheimer's disease uye cognitive impairments.Tsvagiridzo inoratidza kuti Coluracetam inogona kuve neuroprotective zvivakwa, zvichiita kuti ive mumiriri anokatyamadza wekuwedzera kuongororwa mumamiriro aya.Nekudaro, zvimwe zvidzidzo uye miedzo yekiriniki inodiwa kuti uone kushanda kwayo, chengetedzo, uye yakakwana mapuroteni ekushandisa mumakiriniki.

Huwandu hwekuchembera hwakawedzera kudiwa kwekupindira kunogona kudzikisira kuderera kwekuziva kwakabatana nezera.Coluracetam's neuroprotective mhedzisiro uye inogona kutsigira neural kugadzirisa nzira inoita kuti ive nzira inonakidza yekutsvaga mukugadzirisa kuderera kwekuziva kunoenderana nekuchembera.

Uyezve, tsvakurudzo yekutanga inoratidza kuti Coluracetam inogona kuva nemigumisiro yekusagadzikana kwepfungwa zvakadai sekuora mwoyo uye kuzvidya mwoyo.Nekudaro, zvimwe zvidzidzo zvakazara zvinodiwa kuti zviongorore kushanda kwayo uye kumisa nzira dzekurapa dzakakodzera mune izvi zviratidzo.

Simba reColuracetam rinowedzera kune neurorehabilitation zvirongwa zvakare.Kugona kwayo kukwidziridza neuronal kusaina uye inogona kutsigira neural kugadzirisa maitiro inoita kuti ive mumiriri wekushandiswa mukudzoreredza vanhu vane kukuvara kwehuropi kana sitiroko.

Kunyange zvazvo Coluracetam ichiratidza chivimbiso mumashandisirwo akasiyana-siyana, zvakakosha kusimbisa kudiwa kwekuwedzera tsvakurudzo, kusimbisa kushanda kwayo, kuchengeteka, uye kushandiswa kwakakwana kwemitemo.Mvumo yemitemo yaizodiwawo pakushandiswa kwayo kwekiriniki mune chaiyo zviratidzo.


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