Mugadziri weupfu hweColuracetam Nhamba yeCAS: 135463-81-9 99% kuchena kweminiti yezvinongedzo zvekuwedzera
Vhidhiyo yeChigadzirwa
Zvimiro zveChigadzirwa
| Zita rechigadzirwa | Coluracetam |
| Rimwe zita | MKC-231; 2-oxo-N-(5,6,7,8-tetrahydro-2,3-dimethyl-furo[2,3-b]quinolin-4-yl)-1-pyrrolidineacetamide |
| Nhamba yeCAS | 135463-81-9 |
| Fomura yemamorekuru | C19H23N3O3 |
| Kurema kwemasero | 341.4 |
| Kuchena | 99.0% |
| Chitarisiko | Upfu chena |
| Kushandiswa | Zvekudya Zvinowedzerwa Zvekudya Zvakagadzirwa |
Sumo yechigadzirwa
Coluracetam, nhengo yemhuri ye racemate yema nootropic compounds, inozivikanwawo seMKC-231, imushonga we nootropic une simba rekuziva uye kudzivirira tsinga. Coluracetam inoshanda nekugadzirisa cholinergic system. Inofungidzirwa kuti inowedzera huwandu hweacetylcholine, neurotransmitter inokosha muuropi yakabatana zvakanyanya nekudzidza uye mabasa ekurangarira. Coluracetam inoita izvi nekuwedzera huwandu uye basa rezvinhu zvinotakura choline uptake, nokudaro ichisimudzira kuburitswa kweacetylcholine uye kuvandudza masaini pakati pema neuron. Zvimwe zvidzidzo zvekutanga zvekuedza nemhuka zvinoratidza kuti Coluracetam ine simba rekudzivirira tsinga uye kusimudzira tsinga. Zvimwe zvidzidzo zvakawana kuti Coluracetam ine simba rekuvandudza kukanganisa ndangariro muma AD models.
Chinhu
(1) Kuchena kwakanyanya: Coluracetam inogadzirwa uchishandisa nzira dzepamusoro dzekubvisa nekugadzira kuti ive nechokwadi chekuti yakachena kwazvo. Kuchena uku kwakanyanya kunobatsira kuvandudza kuwanikwa kwemishonga uye kuderedza kuitika kwemigumisiro yakaipa.
(2) Kuchengeteka: Coluracetam inoonekwa seyakachengeteka kuvanhu. Zvidzidzo zvakawanda zvakaratidza kuti ine chepfu shoma uye migumisiro mishoma mukati mehuwandu hunokurudzirwa hwemushonga.
(3) Kugadzikana: Mishonga yeColuracetam inoratidza kugadzikana kwakanaka uye inogona kuchengetedza kushanda kwayo uye kushanda kwayo munzvimbo dzakasiyana-siyana nemamiriro ekuchengetedza. Kugadzikana uku kunovimbisa kushanda kwakasimba uye kwakavimbika kwenguva refu.
Mashandisirwo
Coluracetam parizvino inoshandiswa mumhando dzakasiyana siyana uye inoratidza tarisiro huru mune ramangwana. Inonyanya kushandiswa sechikafu chinowedzera kugona kwekufunga uye inotsvakwa nevanhu vari kutsvaga kuvandudza ndangariro, kuisa pfungwa, uye kugona kudzidza. Kugona kwemushonga uyu kugadzirisa system yecholinergic kunofungidzirwa kuti kunobatsira mukuita kwayo kusimudzira kugona kwekufunga. Pamusoro pezvo, tsvakiridzo inoratidza kuti Coluracetam inogona kunge iine hunhu hwekudzivirira tsinga dzinogona kubatsira kudzivirira kudzikira kwekuziva kunokonzerwa nekukwegura uye kutsigira hutano hwehuropi hwese.












