peji_bhena

chigadzirwa

Mugadziri weupfu hweSunifiram Nhamba yeCAS: 314728-85-3 99% kuchena kwezvishandiso zvekuwedzera

Tsananguro pfupi:

Sunifiram mushonga weAMPA receptor agonist unowedzera masaini kubva kumaAMPA receptors muuropi, ayo anowanzo fungidzirwa kuti ndiwo anonyanya kubatsira mukudzidza nekurangarira.


Ruzivo rweChigadzirwa

Matagi eChigadzirwa

Vhidhiyo yeChigadzirwa

Zvimiro zveChigadzirwa

Zita rechigadzirwa

Sunifiram

Rimwe zita

1-(4-Benzoylpiperazin-1-yl)propan-1-one; 1-Benzoyl-4-(1-oxopropyl)piperazine

Nhamba yeCAS

314728-85-3

Fomura yemamorekuru

C14H18N2O2

Kurema kwemasero

246.30

Kuchena

99.0%

Chitarisiko

upfu chena hwekristaro

Kurongedza

1kg/bhegi

Kushandiswa

mishonga ye nootropic

Sumo yechigadzirwa

Sunifiram mushonga weAMPA receptor agonist unowedzera masaini paAMPA receptors muuropi, ayo anowanzo fungidzirwa kuti ane basa guru mukudzidza nekurangarira. Nekuvandudza mashandiro emaAMPA receptors, Sunifiram inofungidzirwa kuti inovandudza kugona kweuropi kudzidza nekurangarira, ukuwo ichivandudzawo kutarisisa uye simba repfungwa. Pamusoro pezvo, inoshanda nekukurudzira mashandiro emaglutamate receptors uye kuwedzera kugadzirwa nekuburitswa kwe "learning neurotransmitter" acetylcholine. Sunifiram inoshanda zvakanyanya seampa factor, zvichireva kuti inosunga kumaAMPA-type glutamate receptors muuropi mushure mekuyambuka chipingamupinyi cheropa-uropi. Izvi zvinokurudzira kugadzirwa kweglutamate, neurotransmitter inokosha yakakosha pa synaptic plasticity, kana kugona kwe nerve synapses kupindura kuwedzera kana kudzikira kwekushanda. Mazinga eGlutamate akakosha zvakanyanya mu hippocampus, chikamu cheuropi chinoita basa rakakosha mukufamba kwenzvimbo, kuumbwa kwendangariro, uye kuchengetwa. Mazinga eglutamate akakwana akakosha pakuwedzera kwenguva refu kana kuvandudzwa kwenguva refu kwemasaini pakati pema neuron. Simba rakakosha. Masimba mazhinji eSunifilaram anowedzera kugona kwepfungwa anoshanda nekuwedzera simba rezviratidzo zvetsinga muchikamu ichi cheuropi.

Chinhu

(1) Kuchena kwakanyanya: Sunifiram inogona kuwana zvigadzirwa zvakachena zvakanyanya kuburikidza nemaitiro ekugadzira akacheneswa. Kuchena kwakanyanya kunoreva kuwanikwa kuri nani kwemuviri uye kushomeka kwemhedzisiro yakaipa.

(2) Kuchengetedzeka: Sunifiram yakaratidzwa kuti haina njodzi kumuviri wemunhu.

(3) Kugadzikana: Sunifiram ine kugadzikana kwakanaka uye inogona kuchengetedza kushanda kwayo uye kushanda kwayo pasi pemamiriro akasiyana-siyana uye mamiriro ekuchengetedza.

Mashandisirwo

Sunifiram mushonga unosimudzira mashandiro etsinga dzemuviri, unowanikwawo sechikafu chinovaka muviri, unofungidzirwa kuti unovandudza mashandiro epfungwa uye unovandudza kudzidza nekurangarira. Unoshanda nekugadzira maAMPA receptors muuropi. AMPA ineurotransmitter inobatsira mukukurukurirana nekukurumidza pakati pemasero ari mutsinga. Inovandudza zvikuru kukurumidza kwekudzidza, kuchengetedza ndangariro nekurangarira, pamwe nekuvandudza kutarisisa, kukurudzira uye kujeka kwepfungwa.


  • Yakapfuura:
  • Zvinotevera:

  • Nyora meseji yako pano woitumira kwatiri