Mugadziri weupfu wePRL-8-53 Nhamba yeCAS: 51352-87-5 98% kuchena kweminiti yezvinongedzo zvekuwedzera
Zvimiro zveChigadzirwa
| Zita rechigadzirwa | PRL-8-53 |
| Rimwe zita | Methyl 3-(2-(benzyl(Methyl)aMino)ethyl)benzoate hydrochloride;Benzoic acid, 3-[2-[methyl(phenylmethyl)amino]ethyl]-, methyl ester, hydrochloride (1:1);Methyl 3-{2-[benzyl(methyl)amino]ethyl}benzoate hydrochloride (1:1) |
| Nhamba yeCAS | 51352-87-5 |
| Fomura yemamorekuru | C18H22ClNO2 |
| Kurema kwemasero | 319.83 |
| Kuchena | 98.0% |
| Chitarisiko | Upfu chena |
| Kurongedza | 1 kg pabhegi rimwe nerimwe 25kg/dhiramu |
| Kushandiswa | nootropic |
Sumo yechigadzirwa
PRL-8-53, inozivikanwawo semethyl 3-(2-(benzyl(methyl)amino)ethyl)benzoate, chinhu chinogadzirwa ne nootropic chinofungidzirwa kuti chinowedzera kutapurirana kwe cholinergic uye Chinodzora huwandu hwe dopamine muuropi. Maitiro aya anobatsira mumhedzisiro yayo inogona kuwedzera kugona kwekuziva, nokudaro ichivandudza kuumbwa kwendangariro, kuchengetedza, uye kudzoreredza. Zvidzidzo zvakawanda pamhuka nevanhu zvakashuma mhedzisiro yakanaka yehunhu hwayo hwekuvandudza ndangariro. Muchidzidzo chekuongorora che double-blind, chakadzorwa ne placebo, vanhu vakagamuchira dose imwe chete yePRL-8-53 vakaratidza kugona kuri nani kwekurangarira mazwi uye kudzoreredza zvichienzaniswa neboka re placebo. Izvi zvakakonzera kufarira uye kutsvagurudza kwakawedzerwa pamusoro pesimba rekomputa. Imwe ongororo mumakonzo yakaratidza kuti kupa PRL-8-53 kwakavandudza zvakanyanya kugona kwavo kudzidza mubasa re water maze. Makonzo akarapwa nePRL-8-53 akakwanisa kuwana puratifomu yakavanzika zviri nani kupfuura kudzora, zvichiratidza kugona kwekomputa sekuwedzera ndangariro.
Chinhu
(1) Kuchena kwakanyanya: PRL-8-53 inogona kuwana zvigadzirwa zvakachena zvakanyanya kuburikidza nemaitiro ekugadzira akacheneswa. Kuchena kwakanyanya kunoreva kuwanikwa kuri nani kwehupenyu uye kushomeka kwemhedzisiro yakaipa.
(2) Kuchengetedzeka: Kuchengeteka kwakanyanya, kusawirirana kushoma, kusawirirana kuri pachena.
(3) Kugadzikana: PRL-8-53 ine kugadzikana kwakanaka uye inogona kuchengetedza kushanda kwayo uye kushanda kwayo pasi pemamiriro akasiyana-siyana uye mamiriro ekuchengetedza.
Mashandisirwo
Semhando itsva yekuwedzera kugona kwepfungwa, PRL-8-53 inovandudza ndangariro yenguva pfupi uye ndangariro yekushanda, ukuwo ichivandudza kugona kwekudzidza uye kukurumidza kuwana hunyanzvi, zvichibatsira kuvandudza kudzidza nekushanda zvakanaka. Tsvagiridzo inoratidza kuti PRL-8-53 inogona kukurudzira kukura nekuvandudzwa kwema neuron muuropi. PRL-8-53 inogona kuwedzera kumhanya uko uropi hunoshandisa ruzivo, zvichibvumira vanhu kupedzisa mabasa uye kuita sarudzo nekukurumidza. Kunyangwe ichienzaniswa nemamwe ma nootropic compounds Zvisinei, tsvagiridzo paPRL-8-53 yakaganhurirwa, asi tsvagiridzo iripo inoratidza kugona kwayo mukuvandudza kugona kwekurangarira nekuziva.











