YDL223C (HBT1) mugadziri wehupfu CAS Nhamba: 489408-02-8 99% kuchena min.zvekuwedzera zvinhu
Product Parameters
Product name | HBT1 |
Rimwe zita | YDL223C |
CAS Nha. | 489408-02-8 |
Molecular formula | C16H17F3N4O2S |
Molecular uremu | 386.40 |
Kuchena | 99.0% |
Chitarisiko | Chiedza chero chakasimba |
Packing | 1kg pabhegi 25kg padhiramu |
Application | nootropics |
Product sumo
HBT1 inosungira kune ligand-binding domain ye-α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor (AMPA-R) nenzira inotenderera-glutamate.Izvi zvinoreva kuti HBT1 imorekuru rinokwanisa kungosunga kune chaiwo masaiti epuroteni yeAMPA-R kana glutamate iripo, uye kuti kusunga uku kunobatsira kuronga kuita kweprotein.AMPA receptors inoratidzwa mukati mepakati tsinga sisitimu uye inoita basa rakakosha mukutaurirana neuronal, kugadzirisa manzwiro, uye kudzidza, ndangariro, uye synaptic plasticity.AMPA receptors ndiwo anobatsira zvikuru mukunakidza neurotransmission, kupindira nekukurumidza, nekukurumidza desensitized kunakidzwa kweakawanda synapses, uye inobatanidzwa mumhinduro dzekutanga dzenzvimbo dzesynaptic kune glutamate.AMPA receptors anowanzo kubatanidzwa neNMDA receptors pamasynapses, uye pamwe chete vanosimudzira synaptic plasticity maitiro anobatanidzwa mukudzidza, ndangariro, excitotoxicity, uye neuroprotection.
Feature
Brain-derived neurotrophic factor (BDNF) is a neurotrophic factor inoita basa rakakosha mukuchengetedza nekuwedzera kweneuroni, uye ine zvine simba uye zvakawanda zvinokonzeresa pakuwanda, kusiyanisa, kurarama uye kufa kwemasero neuronal uye asiri-neuronal, Mabasa se neurotransmitter modulator uye inobatsira kune neuronal plasticity yekudzidza nekuyeuka.Saka zvakakosha kune hutano uye hutano hwenheyo system.Kuwedzera kweBDNF kunogona kuratidza kubatsira mukurapa nekudzivirira kwezvirwere zvakawanda.
Applications
HBT1 inyowani AMPA receptor enhancer ine agonism yakaderera kana ichienzaniswa neLY451395 uye OXP1, inokonzeresa kugadzirwa kwebrain-derived neurotrophic factor (BDNF), uye inoratidza zvishoma mhedzisiro muprimary neurons Agitation.HBT1 inosungira kune ligand-binding domain ye AMPA-R nenzira inotsamira paglutamate.Pamwe chete, vanosimudzira synaptic plasticity maitiro anobatanidzwa mukudzidza, ndangariro, kufara uye neuroprotection.Inogona kuvandudza kugona kwekuziva uye kurangarira kwehuropi, uye kuwedzera kugona kwevanhu kudzidza.