Galantamine Hydrobromide poda inogadzira CAS Nhamba: 1953-04-4 98% kuchena min.zvekuwedzera zvinhu
Product Parameters
Product name | Galantamine Hydrobromide |
Rimwe zita | Galanthamine hydrobromide; Galantamine HBr; Galanthamine HBr;(4aS,6R,8aS)-4a,5,9,10,11,12-hexahydro-3-methoxy-11-methyl-6H-Benzofuro[3a,3,2-ef][2]benzazepin- 6-ol, Hydrobromide |
CAS Nha. | 1953-04-4 |
Molecular formula | C17H21NO3.HBr |
Molecular uremu | 368.27 |
Kuchena | 98.0% |
Chitarisiko | chena kusvika kuchena-upfu |
Packing | 1kg/bag 10kgs,25kgs/drum |
Application | nootropics |
Product sumo
Galantamine hydrobromide imhando ye benzozepine inotorwa kubva kuma bulbs nemaruva e narcissus, osmanthus, kana canna.Iyo zvakare yemuromo cholinesterase inhibitor.Se ligand ye nicotinic acetylcholine receptor, yakashandiswa zvakanyanya kuwedzera neurocognitive basa.Basa rayo nderekukwikwidza uye kudzoreredza kurambidza acetylcholinesterase, nekudaro ichiwedzera kuwanda kweacetylcholine.
Kana yakanyura muropa, galanthamine hydrobromide inotorwa nyore nyore munzvimbo dzese dzemuviri, kusanganisira uropi.Inosungira kune nicotinic acetylcholine receptor, zvichiita kuti conformational shanduko uye kuwedzera acetylcholine kusunungurwa.Inoshandawo nekukwikwidza uye kudzosera mhedzisiro yecholinesterase inhibitors.Nekudzivisa cholinesterase, inodzivirira kuparara kweacetylcholine, nokudaro kuwedzera chiyero uye nguva yeiyi ine simba neurotransmitter.Galanthamine inovandudzawo kudzidza uye kugona kuyeuka, inodzivirira kuzvimba kwehuropi uye inochengetedza yakakwira mazinga eeurotransmitters nekuchengetedza kutendeseka kwemaneuroni uye synapses.
Feature
(1) Imwe mhedzisiro yakakosha yegalanthamine hydrobromide pakuvandudza ndangariro kugona kwayo kuwedzera ndangariro basa.Inowedzera kukurumidza kwekugadzirwa kwendangariro uye inovandudza kuchengetwa kweruzivo uye chokwadi.
(2) Kugona kudzidza kunovandudzwa nekuwedzera synaptic plasticity uye neuroplasticity.Galanthamine hydrobromide zvakananga kana zvisina kunanga inokanganisa neuroplasticity.Inosimudzira synaptic plasticity ne activating microglia uye astrocyte.
(3) Inobatsira kurara uye inowedzera kuzorora.Galanthamine inogona kuwedzera kuoma kwechiitiko chekurara nekukonzera kukurumidza kwekukurumidza kwekufamba kwemaziso kurara, nekudaro kunatsiridza kunaka kwekurara.
(4) Enhance antioxidant dziviriro, Galantamine inopa antioxidant kudzivirira kurwisa oxidative kusagadzikana kunokonzerwa nemahara radicals.Inogona kudzivirira masero ehuropi kubva mukukuvadzwa kweoxidative kuchengetedza yakakwana yehuropi kushanda.