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Galantamine Hydrobromide poda inogadzira CAS Nhamba: 1953-04-4 98% kuchena min.zvekuwedzera zvinhu

Tsanangudzo Pfupi

Imhando ye benzozepine inotorwa kubva kuma bulbs nemaruva e narcissus, osmanthus, kana canna.Iyo zvakare yemuromo cholinesterase inhibitor.


Product Detail

Product Tags

Product Parameters

Product name Galantamine Hydrobromide
Rimwe zita Galanthamine hydrobromide;

Galantamine HBr;

Galanthamine HBr;(4aS,6R,8aS)-4a,5,9,10,11,12-hexahydro-3-methoxy-11-methyl-6H-Benzofuro[3a,3,2-ef][2]benzazepin- 6-ol, Hydrobromide

CAS Nha. 1953-04-4
Molecular formula C17H21NO3.HBr
Molecular uremu 368.27
Kuchena 98.0%
Chitarisiko chena kusvika kuchena-upfu
Packing 1kg/bag 10kgs,25kgs/drum
Application nootropics

Product sumo

Galantamine hydrobromide imhando ye benzozepine inotorwa kubva kuma bulbs nemaruva e narcissus, osmanthus, kana canna.Iyo zvakare yemuromo cholinesterase inhibitor.Se ligand ye nicotinic acetylcholine receptor, yakashandiswa zvakanyanya kuwedzera neurocognitive basa.Basa rayo nderekukwikwidza uye kudzoreredza kurambidza acetylcholinesterase, nekudaro ichiwedzera kuwanda kweacetylcholine.

Kana yakanyura muropa, galanthamine hydrobromide inotorwa nyore nyore munzvimbo dzese dzemuviri, kusanganisira uropi.Inosungira kune nicotinic acetylcholine receptor, zvichiita kuti conformational shanduko uye kuwedzera acetylcholine kusunungurwa.Inoshandawo nekukwikwidza uye kudzosera mhedzisiro yecholinesterase inhibitors.Nekudzivisa cholinesterase, inodzivirira kuparara kweacetylcholine, nokudaro kuwedzera chiyero uye nguva yeiyi ine simba neurotransmitter.Galanthamine inovandudzawo kudzidza uye kugona kuyeuka, inodzivirira kuzvimba kwehuropi uye inochengetedza yakakwira mazinga eeurotransmitters nekuchengetedza kutendeseka kwemaneuroni uye synapses.

Feature

(1) Imwe mhedzisiro yakakosha yegalanthamine hydrobromide pakuvandudza ndangariro kugona kwayo kuwedzera ndangariro basa.Inowedzera kukurumidza kwekugadzirwa kwendangariro uye inovandudza kuchengetwa kweruzivo uye chokwadi.

(2) Kugona kudzidza kunovandudzwa nekuwedzera synaptic plasticity uye neuroplasticity.Galanthamine hydrobromide zvakananga kana zvisina kunanga inokanganisa neuroplasticity.Inosimudzira synaptic plasticity ne activating microglia uye astrocyte.

(3) Inobatsira kurara uye inowedzera kuzorora.Galanthamine inogona kuwedzera kuoma kwechiitiko chekurara nekukonzera kukurumidza kwekukurumidza kwekufamba kwemaziso kurara, nekudaro kunatsiridza kunaka kwekurara.

(4) Enhance antioxidant dziviriro, Galantamine inopa antioxidant kudzivirira kurwisa oxidative kusagadzikana kunokonzerwa nemahara radicals.Inogona kudzivirira masero ehuropi kubva mukukuvadzwa kweoxidative kuchengetedza yakakwana yehuropi kushanda.

Applications

Galantamine hydrobromide inogona kuvandudza ndangariro, kuziva, uye kugona kuita mabasa ezuva nezuva.Inoshanda nekudzorera kuenzana kwezvimwe zvinhu zvakasikwa (neurotransmitters) muuropi.


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